1. Discovery Yrs 1–4
Identify biological targets, druggable binding sites, and develop screening assays to measure compound activity.
2. Lead Optimization Yrs 2–5
Optimize lead series for ADMET properties, selectivity, potency, and scalable synthesis using PK/PD modeling.
3. Preclinical Yrs 4–6
Conduct GLP toxicology studies, determine in vivo safety, efficacy dose, and prepare IND-enabling packages.
4. Clinical Trial Supply (CTS) Scaleup Yrs 5–13
Scale synthesis from lab to GMP, develop formulations, validate analytical methods, and manage clinical supply chain.
5. Regulatory1 Yrs 5–15
eCTD submission, regulatory review, label negotiation, and post-marketing commitment planning.
6. Phase I Yrs 6–8
First-in-human trials to assess safety, tolerability, MTD, and human PK parameters.
7. Phase II Yrs 8–11
Proof-of-concept efficacy trials to determine optimal dose, biomarkers, and target patient subgroups.
8. Phase III Yrs 10–14
Large-scale pivotal trials to confirm efficacy vs. standard of care and build safety database for regulatory approval.
9. Commercial Scale-Up Yrs 13–16
Process validation at commercial scale (PPQ), tech transfer, serialization, and ERP/MES implementation.
10. Commercial & RWE Yr 15+
Post-launch real-world effectiveness monitoring, pharmacovigilance, market access, and HEOR for payers.